中文名 | GLU-THR-PRO-ASP-CYS-PHE-TRP-LYS-TYR-CYS-VAL(DISULFIDE BRIDGE:CYS5-CYS10) |
英文名 | UROTENSIN II (HUMAN) |
英文别名 | UROTENSIN II (HUMAN) UROTENSIN II (HUMAN) HYDROCHLORIDE GLU-THR-PRO-ASP-CYS-PHE-TRP-LYS-TYR-CYS-VAL H-GLU-THR-PRO-ASP-CYS-PHE-TRP-LYS-TYR-CYS-VAL-OH GLU-THR-PRO-ASP-CYS-PHE-TRP-LYS-TYR-CYS-VAL HYDROCHLORIDE |
CAS | 251293-28-4 |
化学式 | C64H85N13O18S2 |
分子量 | 1388.57 |
存储条件 | -15°C |
外观 | 固体 |
体外研究 | Human Urotensin II (U-II) binds to recombinant human GPR14 with high affinity, and the binding is functionally coupled to calcium mobilization. Human Urotensin II induces concentration-dependent increases in intracellular calcium in a HEK-293 cell line expressing human GPR14 (EC 50 =0:62±0.17 nM, n=6). |
体内研究 | Human Urotensin II (U-II) markedly increases total peripheral resistance in anaesthetized non-human primates, a response associated with profound cardiac contractile dysfunction. |
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